WebNov 28, 2016 · Cytochalasin E ( 57) was the most active compound. It was toxic against brine shrimp with a LC 50 of 2.79 μM, which is comparable to the commercial insecticidal toosendanin (LC 50 = 4.03 μM). Compounds 54 - 55 and 93 showed low toxicity toward brine shrimp, ≤10% mortality at 50 μM (Zhang et al. 2014 ). WebJun 1, 2024 · Here, we obtained cytochalasin Q (CQ) from Xylaria sp. DO1801, the endophytic fungi from the root of plant Damnacanthus officinarum, and discovered its …
Cytotoxic cytochalasans from cultures of the fungus
WebJan 11, 2024 · Here, we use the aspo cluster of aliphatic amino acid-type cytochalasin compounds (aspochalasans) as the research target and demonstrate that (1) reconstitution of the four-gene conserved cassette ... WebSep 10, 2024 · Cytochalasans or “cytochalasins” are macromolecular fungal metabolites displaying significant cytotoxicity. Their complex structures are assembled by hybrid polyketide synthase (PKS)-nonribosomal... imaging assoc of indiana
(PDF) Actin cytoskeletal inhibitor 19,20-epoxycytochalasin Q …
WebAug 6, 2001 · Three known compounds, 2-hexylidene-3-methylsuccinic acid (1), cytochalasin Q (2), and 5-carboxymellein (3), together with two new derivatives, 2-hexylidene-3-methylsuccinic acid 4-methyl ester (4) and an ophiobolane sesterterpene named halorosellinic acid (5), were isolated from culture broth of the marine fungus … WebDihydrocytochalasin B (H2CB) inhibits active calcium transport and causes a Ca 2+ increase in the mucosal scrapings. Cytochalasin B is a cell-permeable mycotoxin binding to the … WebApr 12, 2024 · Optimization of incubation with cytochalasin B in the EpiAirway™ model. a Schematic of the incubation conditions with cytochalasin B (CB) for 48 or 72 h.b Percentage of binucleated cells (%BNCs) obtained after incubation with at 0, 1, 3, and 5 μg/mL for 48 h (in light blue) or 72 h (in blue).c Schematic of the incubation conditions … imaging at foothills hospital boulder co